PTH1R

PTH1R

PTH1R Molekülinformation

Molecule Name
Parathyroid hormone receptor
Molekülalias
PTH1R,PTHR,PTHR1
Drug Development Progress
Anzahl der klinischen Arzneimittel25
Anzahl der inverkehr gebrachten Arzneimittel23
Höchste Forschungs- und EntwicklungsphaseApproved
Target-Alias
Receptors, Parathyroid Hormone
Molekülhintergrund
Parathyroid hormone/parathyroid hormone-related peptide receptor is also known as Parathyroid hormone 1 receptor (PTH1R), PTHR1, PTH/PTHrP type I receptor (PTH/PTHr receptor), which belongs to the G-protein coupled receptor 2 family. PTH1R / PTHR1 is a receptor for parathyroid hormone and for parathyroid hormone-related peptide. The activity of this receptor is mediated by G proteins which activate adenylyl cyclase and also a phosphatidylinositol-calcium second messenger system.

PTH1R Produktliste

Species
  • Human(2)
Tag
  • -(1)
  • His Tag(1)
Host
  • HEK293(2)
Conjugate
  • Unconjugated(2)
Grade
  • RUO(2)
Low Endotoxin
  • Yes(1)
  • No(1)
MoleculeCat. No.Product NameArtHostStructurePurityActivitySize&PriceAdd to Cart
PTH1R
Human PTH1R / PTHR1 Protein, His Tag, low endotoxin (MALS verified)
Human
HEK293
MALSSDS-PAGE
ELISA

$260.00

100ug
PTH1R
Human PTH1R Full Length Protein (VLP)
Human
HEK293
HPLC
ELISAIdentity

$620.00

20ug
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Klinische Arzneimittelinformation

Englischer NameForschungscodeForschungsphaseFirmaIndikationenKlinische Studie
Teriparatide biosimilar (National Institute of Dental and Craniofacial Research)rhPTH (1-34) (National Institute of Dental and Craniofacial Research)Phase 3 ClinicalNational Institute Of Dental And Craniofacial Research
DiGeorge Syndrome; Hypoparathyroidism; Hypothyroidism
Details
Teriparatide biosimilar (Shanghai CAS Shenglongda Biotech)Phase 3 ClinicalShanghai Zhongke Shenglongda Biotechnology (Group) Co Ltd
Osteoporosis, Postmenopausal
Details
Parathyroid hormone 1-84 (Kerun Biopharmaceutical)Phase 3 ClinicalChongqing Kerun Biologic Pharmaceutical Development Co Ltd
Hypoparathyroidism; Osteoporosis, Postmenopausal
Details
MT-1013MT-1013Phase 3 ClinicalShaanxi Micot Pharmaceutical Technology Co Ltd
Hyperparathyroidism; Hyperparathyroidism, Secondary; Renal Insufficiency, Chronic
Details
EneboparatideAZP-3601Phase 3 ClinicalHarvard Medical School, Massachusetts General Hospital
Endocrine System Diseases; Hypoparathyroidism; Parathyroid Diseases
Details
Teriparatide transdermal (Corium International)Phase 2 ClinicalCorium International Inc
Osteoporosis
Details
Teriparatide transdermal (Zosano Pharma)B-106; B-104; ZP-PTH; ThPTH (1-34); TH-0229Phase 2 ClinicalZosano Pharma Corp
Osteoporosis; Osteoporosis, Postmenopausal
Details
KUR-113KUR-113; I-040202; Fibrin-PTHPhase 2 ClinicalKuros Biosciences
Intervertebral Disc Degeneration; Spinal Diseases; Wounds and Injuries
Details
T3-sulfate (Bracco SpA)Phase 2 ClinicalBracco Spa
Hypothyroidism
Details
Recombinant Human Parathyroid Hormone (1-34)(Shanghai Celgen Biopharmaceuticals)Phase 2 ClinicalShanghai Celgen Bio-Pharmaceutical Co Ltd
Osteoporosis
Details
KUR-111I-0401; KUR-111Phase 2 ClinicalKuros Biosciences
Fractures, Bone
Details
ST-1891ST-1891Phase 2 ClinicalSention Therapeutics LLC
Hypothyroidism
Details
Teriparatide oral (Entera Bio)EB612; EB-612; EB-613; PTH 1-34; EBP-05; EBP05; hPTH(1-34) (Entera Bio); PTH-1-34Phase 2 ClinicalEntera Bio Ltd
Drug-Related Side Effects and Adverse Reactions; Fractures, Stress; Hypoparathyroidism; Osteoporosis
Details
EXT-608EXT-608Phase 2 ClinicalExtend Biosciences Inc
Hypoparathyroidism
Details
CanvuparatideMBX-2109; MBX 2109Phase 2 ClinicalMBX Biosciences Inc
Hypoparathyroidism; Renal Insufficiency
Details
Teriparatide biosimilar (Shanghai Fudan-Zhangjiang Bio-Pharmaceutical)Phase 1 ClinicalShanghai Fudan-Zhangjiang Bio-Pharmaceutical Co Ltd
Osteoporosis
Details
HemoparatidehPTH-137Phase 1 ClinicalPharis Biotec
Psoriasis
Details
Tripatide (Yunnan First Applied Pharma)Phase 1 ClinicalYunnan First Applied Pharmaceutical Industry
Osteoporosis
Details
SEP-786SEP-786Phase 1 ClinicalSepterna Inc
Hypoparathyroidism
Details
Teriparatide biosimilar (Shanghai Duomirui)Phase 1 ClinicalShanghai Duomirui Biotechnology Co Ltd
Osteoporosis
Details
Teriparatide biosimilar (Wuxi Hebang)Phase 1 ClinicalWuxi Hebang Biotechnology Co Ltd
Osteoporosis; Osteoporosis, Postmenopausal; Osteoporotic Fractures
Details
RT-102(Rani)RT-102Phase 1 ClinicalRani Therapeutics Holdings Inc
Osteoporosis
Details
Parathyroid hormone 1-84(Sichuan Luzhou Buchang Biopharmaceutical)Phase 1 ClinicalSichuan Luzhou Buchang Biopharmaceutical Co Ltd
Hypocalcemia
Details
MT-1009MT-1009Phase 1 ClinicalShaanxi Micot Pharmaceutical Technology Co Ltd
Glucocorticoid-induced osteoporosis; Osteoporosis
Details
BMD-1221BMD-1221ClinicalUniversity Of Arkansas System
Fractures, Bone
Details

Inverkehr gebrachte Arzneimittelinformation

Englischer NameForschungscodeForschungsphaseFirmaFrühestes MarkennameFrühestes GenehmigungslandFrüheste IndikationFrüheste GenehmigungsgesellschaftFrüheste GenehmigungsdatumIndikationenKlinische Studie
PalopegteriparatideACP-014; ACP014; ACP 014ApprovedAscendis PharmaTransCon, YORVIPATHEUHypoparathyroidismAscendis Pharma Bone Diseases As, Ascendis Pharma2023-11-17
Endocrine System Diseases; Hypoparathyroidism; Parathyroid Diseases
Details
Teriparatide biosimilar (Biosidus)rhPTH (1-34) (Biosidus)ApprovedBiosidusOsteofortilArgentinaOsteoporosisBiosidus2012-08-01
Osteoporosis
Details
Teriparatide biosimilar (Amega Biotech)rhPTH (1-34) (Amega Biotech)ApprovedAmega Biotech
Osteoporosis
Details
Teriparatide biosimilar (Pfenex)rhPTH (1-34) (Pfenex); PF-708ApprovedPfenex Biopharmaceuticals IncBonsity, QutavinaUnited StatesGlucocorticoid-induced osteoporosis; Osteoporosis, Postmenopausal; OsteoporosisAlvogen2019-10-04
Glucocorticoid-induced osteoporosis; Osteoporosis; Osteoporosis, Postmenopausal
Details
TeriparatideLY 333334; hPTH-1-34; MN-10TApprovedEli Lilly And CompanyForteo, Forsteo, 复泰奥United StatesOsteoporosisEli Lilly And Company2002-11-26
Ankle Fractures; Anorexia Nervosa; Back Pain; Bone Diseases, Metabolic; Cartilage Diseases; Chronic Kidney Disease-Mineral and Bone Disorder; Colles' Fracture; Femoral Neck Fractures; Fractures, Bone; Humeral Fractures; Hyperparathyroidism, Secondary; Hypocalcemia; Hypoparathyroidism; Menopausal symptoms; Osteoarthritis, Knee; Osteoporosis; Osteoporosis, Postmenopausal; Periodontitis; Spinal Cord Injuries; Spinal Fractures
Details
Parathyroid hormone (Shire)SHP-634; ALX-111; 423562; NPSP-795; rhPTH (1-84); SHP-635; rhPTH-1-84; PTH (1-84); SB-423562; PTH 1-84; NPSP-558ApprovedShireNatpara, Preotact, NatparUnited StatesHypoparathyroidismNps Pharmaceuticals, Inc2006-04-24
Autosomal Dominant Hypocalcemia Type 1; Bone Diseases, Endocrine; Hyperparathyroidism; Hypocalcemia; Hypoparathyroidism; Osteoporosis; Osteoporosis, Postmenopausal; Plaque psoriasis
Details
Teriparatide biosimilar (Intas Pharmaceuticals)rhPTH (1-34) (Intas Pharmaceuticals); INTG8; INTG-8ApprovedIntas BiopharmaceuticalsTerifracIndiaOsteoporosisIntas Biopharmaceuticals2010-12-01
Osteoporosis
Details
Teriparatide biosimilar (Gedeon Richter)rhPTH (1-34) (Gedeon Richter)ApprovedGedeon Richter PlcTerrosaEUOsteoporosisGedeon Richter Plc2017-01-04
Fractures, Stress; Osteoporosis
Details
Teriparatide biosimilar (Salubris)SAL056; G56-W1; SAL-001ApprovedShenzhen Salubris Pharmaceuticals Co Ltd欣复泰Mainland ChinaOsteoporosis, PostmenopausalSuzhou Genemen Biotech Co Ltd2019-09-29
Osteoporosis, Postmenopausal
Details
Teriparatide biosimilar (USV)ApprovedUSV Pvt Ltd
Osteoporosis
Details
Teriparatide biosimilar (Strides Pharma)SBL-001ApprovedStrides PharmaKaulivEUOsteoporosis; Osteoporosis, PostmenopausalStrides Pharma (Cyprus) Ltd2023-01-12
Osteoporosis; Osteoporosis, Postmenopausal
Details
Teriparatide biosimilar (STADA Arzneimittel AG)rhPTH (1-34) (STADA Arzneimittel AG)ApprovedStada Arzneimittel AgMovymiaEUOsteoporosisStada Arzneimittel Ag2017-01-11
Osteoporosis
Details
Teriparatide biosimilar (Teva)ApprovedTevaIrelandOsteoporosisTeva Bv2018-06-22
Osteoporosis
Details
Teriparatide biosimilar (Almaject)ApprovedAlmaject IncUnited StatesOsteoporosis; Osteoporosis, PostmenopausalAlmaject Inc2024-06-04
Osteoporosis; Osteoporosis, Postmenopausal
Details
Recombinant parathyroid hormone biosimilar(Chongqing Fujin Biological Medicine)ApprovedChongqing Fujin Biological Medicine Co Ltd
Details
Recombinant Human Parathyroid Hormone (1-34), Shanghai FosunpharmaApproved
Details
Teriparatide acetatehPTH (1-34) acet. H2O; AK-159; MN-10-TApprovedUnion Square Ventures LlcParathar, TeriboneJapanHypocalcemia; Osteoporosisnull1987-03-31
Hypocalcemia; Osteoporosis
Details
Teriparatide biosimilar (Theramex)ApprovedTheramex Ireland LtdLivogivaEUOsteoporosisTheramex Ireland Ltd2020-08-27
Osteoporosis
Details
Teriparatide biosimilar (Shanghai United Cell )ApprovedShanghai United Cell Biotechnology Co LtdMainland ChinaOsteoporosisShanghai United Cell Biotechnology Co Ltd2017-03-22
Osteoporosis
Details
Teriparatide biosimilar (Beijing Bokangjian Gene)ApprovedBeijing Genetech Pharmaceutical Co Ltd博固泰Mainland ChinaOsteoporosisBeijing Genetech Pharmaceutical Co Ltd2024-01-16
Osteoporosis; Osteoporosis, Postmenopausal
Details
Teriparatide biosimilar (Virchow/Sun)rhPTH (1-34) (Virchow/Sun)ApprovedSun Pharmaceutical Industries Ltd, Virchow GroupBonista, OsteotideEUOsteoporosis; Osteoporosis, PostmenopausalSun Pharmaceutical Industries (Europe) Bv
Osteoporosis; Osteoporosis, Postmenopausal
Details
Teriparatide biosimilar (CinnaGen)rhPTH (1-34) (CinnaGen)ApprovedCinnagenCinnoParIranOsteoporosisCinnagen2013-01-01
Osteoporosis
Details
Teriparatide biosimilar (Zydus Cadila)rhPTH (1-34) (Zydus Cadila)ApprovedZydus CadilaIndiaOsteoporosisZydus Cadila2014-01-01
Osteoporosis
Details
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