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MRGPRX2

MRGPRX2 Produktliste

  • Attribut

    Cell (3)Protein (4)

  • Produktbibliothek

    Online (6)In Forschung (1)

  • Spezies

    Human (7)

  • Etikett

    - (6)Flag Tag & Avi Tag (1)

  • Marker

    - (3)Unconjugated (2)Biotin-labeled (1)FITC Labeled (1)

MRGPRX2 Molekülhintergrund

The protein belongs to the family of G-protein coupled receptors, that are preferentially activated by adenosine and uridine nucleotides. It is moderately expressed in undifferentiated HL60 cells, and is located on both chromosomes X and Y.

Klinische Arzneimittelinformation

Englischer NameForschungscodeForschungsphaseFirmaIndikationenKlinische Studie
Dronabinol(AXIM Biotechnologies)Phase 3 ClinicalAxim BiotechNeoplasms; Child Nutrition Disorders; Vomiting; Nausea; Cachexia; Sarcopenia; Anorexia Nervosa
Details
AdezunapAP-707Phase 3 ClinicalCannaXan GmbHMultiple Sclerosis; Accidental Injuries; Low Back Pain; Diabetes Mellitus; Peripheral Nerve Injuries; Diabetic peripheral neuropathy; Back Pain; Neuralgia; Somatoform Disorders; Stroke; Peripheral Nervous System Diseases; Brachial Plexus Neuropathies; Phantom Limb; Pain, Postoperative; Diabetic Neuropathies; Brain Injuries, Traumatic; Chronic Pain; Pain; Paraplegia
Details
Dronabinol(Vertanical)VER-01Phase 3 ClinicalVertanical GmbHLow Back Pain
Details
cannabidiol (Cardiol Therapeutics)Phase 3 ClinicalCardiol Therapeutics IncCoronavirus Disease 2019 (COVID-19); Pericarditis; Cardiovascular Diseases; Myocarditis
Details
V-24343V-24343; ANEB-001Phase 2 ClinicalVernalis PlcPoisoning; Obesity
Details
11C-MePPEP11C-MePPEPPhase 2 ClinicalEli Lilly And CompanySubstance-Related Disorders; Obesity
Details
AX-1602AX-1602Phase 2 ClinicalAxim BiotechPsoriasis; Dermatitis, Atopic; Vitiligo
Details
NimacimabRYI-018; RYI-028; JNJ-2463Phase 2 ClinicalBird Rock Bio IncMetabolic Dysfunction-Associated Steatotic Liver Disease; Renal Insufficiency, Chronic; Obesity; Diabetic Gastroparesis
Details
ART-2713NEO-1940; ART-2713; ART27.13; AZD-1940Phase 2 ClinicalAstrazeneca Plc, Neomed Inc, Pfizer IncWeight Loss; Pain; Anorexia; Cachexia; Low Back Pain
Details
Cannabidiol/hydroxychloroquineIHL-675A; IHL-675Phase 2 ClinicalIncannex Healthcare LtdArthritis, Rheumatoid; Respiratory Distress Syndrome, Adult
Details
AEF-0217AEF-0217Phase 2 ClinicalAelis FarmaDown Syndrome
Details
MonlunabantMRI-1891; NN9440–INV-202; INV-202Phase 2 ClinicalInversago Pharma IncMetabolic Syndrome; Metabolic Diseases; Diabetic Nephropathies; Obesity
Details
IGC-AD1IGC-AD1Phase 2 ClinicalUniversity Of South FloridaAnxiety; Depression; Alzheimer Disease; Psychomotor Agitation; Memory Disorders
Details
AEF-0117AEF-0117Phase 2 ClinicalNational Institute On Drug Abuse, Aelis FarmaMarijuana Abuse
Details
[11C]OMAR[11C]JHU-75528Phase 1 ClinicalJohns Hopkins University School Of MedicineMarijuana Abuse; Schizophrenia
Details
ZYN-001ZYN-001Phase 1 ClinicalZynerba PharmaceuticalsNeuralgia; Fibromyalgia
Details
TetrahydrocannabivarinGWP-42004; THCV; O-4394; DELTA9-THCV; GW-42004Phase 1 ClinicalGw Pharmaceuticals PlcDiabetes Mellitus, Type 2; Hyperglycemia; Metabolic Syndrome; Obesity, Morbid; Hypercholesterolemia; Dyslipidemias
Details
ZevaquenabantMRI-1867; (S)-MRI-1867; INV-101Phase 1 ClinicalNational Institutes Of HealthScleroderma, Systemic; Colitis, Ulcerative
Details
TPT0301TPT-0301; TPT0301Phase 1 ClinicalTetra Pharm Technologies ApSChronic Pain
Details
INV-347NN9441; NN-9441; INV-347Phase 1 ClinicalInversago Pharma IncObesity
Details
IPI 201(Isosceles Pharmaceuticals Inc )IPI-201Phase 1 ClinicalPain, Postoperative
Details
GFB-024Phase 1 ClinicalTakeda PharmaKidney Diseases; Endocrine System Diseases; Diabetic Nephropathies; Diabetes Complications; Diabetes Mellitus
Details
DBPR-211Phase 1 ClinicalNational Health Research InstitutesDiabetes Mellitus, Type 2
Details
MP-10XMP-10XClinicalMedipure HoldingsPain
Details
Cannabidiol/PalmitoylethanolamideTHX-210; SCI–210ClinicalTherapix Biosciences LtdAutism Spectrum Disorder; Diabetic Neuropathies
Details
C20T5C20T5Murdoch Childrens Research Institute
Details
C12T12C12T12Murdoch Childrens Research Institute
Details

Inverkehr gebrachte Arzneimittelinformation

Englischer NameForschungscodeForschungsphaseFirmaFrühestes MarkennameFrühestes GenehmigungslandFrüheste IndikationFrüheste GenehmigungsgesellschaftFrüheste GenehmigungsdatumIndikationenKlinische Studie
Cannabidiol/DronabinolTHC-5; delta-9-THC/CBD; MPL-001; MPL-005; GW-1000; KL16-012; BOL-DP-o-04; GW-1000-02; PPP-001; MGC-ODTApprovedGw PharmaceuticalsSativex, QixleefCanadaMuscle Spasticity; Neuralgia; Cancer Pain; Chronic Pain; Multiple Sclerosisnull2005-04-01Back Pain; Phobia, Social; Neuralgia, Postherpetic; Huntington Disease; Reflex Sympathetic Dystrophy; Tourette Syndrome; Muscle Spasticity; Malnutrition; Sciatica; Acute Pain; Neuromyelitis Optica; Arthritis, Psoriatic; Neuralgia; Dementia; Panic Disorder; Osteoarthritis, Knee; Hepatic Insufficiency; Stress Disorders, Post-Traumatic; Healthy Aging; Hidradenitis Suppurativa; Agoraphobia; Drug Resistant Epilepsy; Renal Insufficiency, Chronic; Social Behavior; Corticobasal degeneration; Cerebral Palsy; Low Back Pain; Neoplasms; Sleep Initiation and Maintenance Disorders; Peripheral Nervous System Diseases; Pain; Chronic Pain; Depression; Depressive Disorder, Major; Marijuana Abuse; Marijuana Use; Spasm; Squamous Cell Carcinoma of Head and Neck; Cancer Pain; Renal Insufficiency; Spinal Cord Injuries; Migraine Disorders; Arthritis, Rheumatoid; Neck Pain; Diabetic Neuropathies; Sleep Wake Disorders; Opioid-Related Disorders; Essential Tremor; Anorexia; Anxiety Disorders; Kidney Diseases; Multiple Sclerosis; Tic Dis
Details
CannabidiolAVCN-583601; GLA-015; BTX-1503; BTX-1801; BTX-1702; LYT-310; RAD011; PBX-1308; RAD-011; BRCX-014; RLS-103; GWP-42003; GWP-42003-P; BOL-DP-o-05; GW-42003; BTX-1204; ZYN-002; PTL-101; CHI-902; APH-1501ApprovedGw Pharmaceuticals PlcEpidiolex, Epidyolex, Zygel, CannepilUnited StatesEpilepsies, Myoclonic; Lennox Gastaut Syndromenull2018-06-25Migraine Disorders; Peripheral Nervous System Diseases; Acne Vulgaris; HIV Infections; Tobacco Smoking; Ovarian Neoplasms; Sleep Initiation and Maintenance Disorders; Facial Pain; Substance-Related Disorders; Marijuana Smoking; Tobacco Use Cessation; Anxiety; Pain; Chronic Pain; Marijuana Use; Seizures; Tuberous Sclerosis; Rett Syndrome; Schizophrenia; Appetitive Behavior; Autism Spectrum Disorder; Marijuana Abuse; Brain Injuries, Traumatic; Depression; Alcoholic Intoxication; Inflammatory Bowel Diseases; Fatty Liver; Child Behavior Disorders; Diabetes Mellitus, Type 2; Spinal Cord Injuries; Sleep Wake Disorders; Anxiety Disorders; Neoplasms; Opioid-Related Disorders; Diabetic Neuropathies; Coronavirus Disease 2019 (COVID-19); Musculoskeletal Pain; Graft vs Host Disease; Blepharospasm; Dyspepsia; Arthritis, Rheumatoid; Psychotic Disorders; Hyperalgesia; Chronic Urticaria; Hoarding Disorder; Bipolar Disorder; Pancreatic Neoplasms; Brain Diseases; Dysmenorrhea; Sturge-Weber Syndrome; Lennox Gastaut Syndrome; Ph
Details
  • Produktliste
  • Inverkehr gebrachte Arzneimittelinformation
  • Klinische Arzneimittelinformation
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