ADORA2A

ADORA2A

ADORA2A Molekülinformation

Molecule Name
Adenosine A2a receptor
Molekülalias
ADORA2A,adenosine A2a receptor,A2aR, ADORA2, RDC8
Drug Development Progress
Anzahl der klinischen Arzneimittel23
Anzahl der inverkehr gebrachten Arzneimittel53
Höchste Forschungs- und EntwicklungsphaseApproved
Target-Alias
Adenosine receptor A2a,ADORA2A,Adenosine A2a Receptor,ADORA2,Adenosine Receptor Subtype A2a,A2aR,RDC8,Receptor, Adenosine A2A
Molekülhintergrund
Adenosine Receptor Subtype A2a (ADORA2A) is a G-protein coupled adenosine receptor encoded by the ADORA2A gene. It is mainly involved in pathophysiological processes including neuroinflammation, synaptic plasticity in glutamatergic synapses and neurogenesis.

ADORA2A Produktliste

Species
  • Human(2)
Tag
  • -(1)
  • His Tag & Flag Tag(1)
Host
  • HEK293(2)
Conjugate
  • Unconjugated(2)
Grade
  • RUO(2)
Low Endotoxin
  • No(2)
MoleculeCat. No.Product NameArtHostStructurePurityActivitySize&PriceAdd to Cart
ADORA2A
Human ADORA2A Protein, Flag,His Tag (Detergent)
Human
HEK293
SDS-PAGE
ELISA

$805.00

20ug
ADORA2A
Human ADORA2A Full Length Protein (VLP)
Human
HEK293
HPLC
ELISAIdentity

$620.00

20ug
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Klinische Arzneimittelinformation

Englischer NameForschungscodeForschungsphaseFirmaIndikationenKlinische Studie
Naproxen/CaffeineBAY-2880376Phase 3 ClinicalBayer AG
Pain, Postoperative
Details
ImaradenantAZD-4635; HTL-1071Phase 2 ClinicalNxera Pharma UK Ltd
Carcinoma, Non-Small-Cell Lung; Colorectal Neoplasms; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Solid tumours
Details
CiforadenantCPI-444; V-81444Phase 2 ClinicalVernalis (R&D) Ltd
Attention Deficit Disorder with Hyperactivity; Carcinoma, Non-Small-Cell Lung; Carcinoma, Renal Cell; Multiple Myeloma; Neoplasms; Parkinson Disease
Details
CaffeinolPhase 2 ClinicalCardium Therapeutics
Alcoholic Intoxication; Alcoholism; Carcinoma, Non-Small-Cell Lung; Disruptive, Impulse Control, and Conduct Disorders; Ischemic Stroke
Details
EtrumadenantAB-928; GS-0928Phase 2 ClinicalArcus Biosciences Inc
Breast Neoplasms; Carcinoma, Merkel Cell; Carcinoma, Non-Small-Cell Lung; Carcinoma, Pancreatic Ductal; Carcinoma, Renal Cell; Carcinoma, Squamous Cell; Carcinoma, Transitional Cell; Colorectal Neoplasms; Endometrial Neoplasms; Esophageal Neoplasms; Head and Neck Neoplasms; Hormone-Resistant Prostate Neoplasms; Hypopharyngeal Neoplasms; Laryngeal Neoplasms; Lung Neoplasms; Melanoma; Mouth Neoplasms; Neoplasm Metastasis; Oral Squamous Cell Carcinoma; Oropharyngeal Neoplasms; Oropharyngeal Squamous Cell Carcinoma (OPSCC); Ovarian Neoplasms; Pharyngeal Neoplasms; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Rectal Neoplasms; Squamous Cell Carcinoma of Head and Neck; Stomach Neoplasms; Triple Negative Breast Neoplasms; Urinary Bladder Neoplasms
Details
PORT-8PORT-8; TT-53Phase 2 ClinicalTarus Therapeutics Inc
Solid tumours
Details
ND10(Theialife Inc)ND-10; ND10Phase 2 ClinicalTheialife Inc
Cataract; Dry Eye Syndromes; Myopia
Details
PORT-6PORT-6; TT-10Phase 2 ClinicalImpetis Biosciences Ltd
Carcinoma, Non-Small-Cell Lung; Carcinoma, Renal Cell; Colorectal Neoplasms; Endometrial Neoplasms; Neoplasms; Ovarian Neoplasms; Prostatic Neoplasms, Castration-Resistant; Squamous Cell Carcinoma of Head and Neck
Details
MK-1088MK-1088Phase 2 ClinicalMerck Sharp & Dohme LLC
Solid tumours
Details
VG081821ACVG081821AC; VG-081821ACPhase 2 ClinicalZhejiang Vimgreen Pharmaceuticals Ltd
Metabolic Dysfunction-Associated Steatotic Liver Disease; Parkinson Disease
Details
ILB-2109WTS-001; ILB-2109Phase 2 ClinicalHangzhou Wutong Tree Pharmaceutical Co Ltd
Carcinoma, Non-Small-Cell Lung; Endometrial Neoplasms; Head and Neck Neoplasms; Hodgkin Disease; Melanoma; Nasopharyngeal Carcinoma; Neoplasms; Ovarian Neoplasms; Sarcoma; Solid tumours; Triple Negative Breast Neoplasms; Uterine Cervical Neoplasms
Details
PBF-999PBF-999Phase 1 ClinicalPalobiofarma Sl
Huntington Disease; Neoplasms
Details
[18F]MNI-444[18F]MNI-444Phase 1 ClinicalInvicro Llc
Diagnostic agents
Details
SHR-5126SHR-5126Phase 1 ClinicalJiangsu Hengrui Medicine Co Ltd
Neoplasms
Details
TaminadenantNIR-178; PBF-509Phase 1 ClinicalPalobiofarma Sl
Carcinoma; Carcinoma, Non-Small-Cell Lung; Carcinoma, Pancreatic Ductal; Carcinoma, Renal Cell; Colorectal Neoplasms; Head and Neck Neoplasms; Lymphoma, Large B-Cell, Diffuse; Melanoma; Ovarian Neoplasms; Pancreatic Neoplasms; Parkinson Disease; Prostatic Neoplasms, Castration-Resistant; Solid tumours; Triple Negative Breast Neoplasms
Details
ST-4206ST-4206Phase 1 ClinicalAlfasigma Spa
Parkinson Disease
Details
CKD-512CKD-512Phase 1 ClinicalChong Kun Dang Pharmaceutical Corp
Neoplasms; Solid tumours
Details
JNJ-86974680JNJ-86974680Phase 1 ClinicalJohnson & Johnson Enterprise Innovation Inc
Carcinoma, Non-Small-Cell Lung; Prostatic Neoplasms
Details
YZJ-5053YZJ5053; YZJ-5053Phase 1 ClinicalShanghai Haiyan Pharmaceutical Technology Co Ltd
Neoplasm Metastasis; Solid tumours
Details
CT-1500CT-1500Phase 1 ClinicalCircadian Technologies Ltd
Details
DZD-2269DZD-2269Phase 1 ClinicalDizal Pharmaceutical Co Ltd
Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant
Details
INCB-106385INCB-106385Phase 1 ClinicalIncyte Corp
Carcinoma, Hepatocellular; Carcinoma, Non-Small-Cell Lung; Carcinoma, Pancreatic Ductal; Colorectal Neoplasms; Gastrointestinal Neoplasms; Ovarian Neoplasms; Prostatic Neoplasms, Castration-Resistant; Solid tumours; Squamous Cell Carcinoma of Head and Neck; Triple Negative Breast Neoplasms; Urinary Bladder Neoplasms
Details
CS-3005CS-3005Phase 1 ClinicalCstone Pharmaceuticals (Suzhou) Co Ltd
Solid tumours
Details

Inverkehr gebrachte Arzneimittelinformation

Englischer NameForschungscodeForschungsphaseFirmaFrühestes MarkennameFrühestes GenehmigungslandFrüheste IndikationFrüheste GenehmigungsgesellschaftFrüheste GenehmigungsdatumIndikationenKlinische Studie
Regadenoson HydrateCVT-3146ApprovedAstellas Pharma IncRapiscan, 海诺生, LexiscanUnited StatesContrast agentsAstellas Pharma Inc2008-04-10
Anemia, Sickle Cell; Astrocytoma; Cardiovascular contrast agents; Cardiovascular Diseases; Contrast agents; Coronary Artery Disease; Coronavirus Disease 2019 (COVID-19); Diagnostic agents; Glioblastoma; Glioma; Heart Diseases; Myocardial Ischemia; Oligodendroglioma; Pneumonia; Rejection of lung transplantation; Retinal Artery Occlusion
Details
Caffeine/Ergotamine TartrateApprovedNovartis Pharma AgCafergotJapanVascular Headaches; Migraine Disorders; Tension-Type HeadacheNichi-Iko Pharmaceutical Co Ltd1948-11-26
Migraine Disorders; Tension-Type Headache; Vascular Headaches
Details
OxtriphyllineApprovedTheocolinCanadanull
Asthma
Details
Caffeine/Metamizole Sodium/Dihydroergotamine MesylateApprovedCefaliv
Migraine Disorders
Details
AdenineApprovedLeuconJapanLeukopeniaOhara Pharmaceutical Co Ltd
Leukemia; Leukopenia
Details
Acetaminophen/Butalbital/Caffeine/Codeine PhosphateApprovedActavis Laboratories Ut IncUnited StatesHeadache; Headache DisordersActavis Laboratories Ut Inc1992-07-30
Headache; Headache Disorders
Details
IstradefyllineKW-6002ApprovedKyowa Hakko Kirin Co LtdNourianz, NouriastJapanParkinson DiseaseKyowa Hakko Kirin Co Ltd2013-03-25
Amyotrophic Lateral Sclerosis; Cognition Disorders; Hepatic Insufficiency; Movement Disorders; Parkinson Disease; Restless Legs Syndrome; Sleep Wake Disorders; Substance-Related Disorders
Details
Sodium Citrate/Citric Acid/Dextrose/Monosodium phosphate/Adenine/Mannitol/Sodium ChlorideApproved
Details
Sodium Citrate/Citric Acid/DextroseApproved
Details
Sodium Citrate/Citric Acid/Dextrose/Monosodium phosphate/AdenineApproved
Details
Aspirin/Acetaminophen/Caffeine/ThiamineApproved
Fever; Pain
Details
Propranolol hydrochloride/Caffeine/Phenytoin SodiumApprovedMainland ChinaHebei Tiancheng Pharmaceutical Co Ltd
Details
Salicylamide/Acetaminophen/CaffeineApproved
Arthralgia; Fever; Headache; Neuralgia; Rheumatic Diseases
Details
Compound Paracetamol Caffeine and Pseudoephedrine HydrochlorideApproved
Common Cold
Details
Acetaminophen/Methylephedrine Hydrochloride/Dextromethorphan Hydrobromide/Chlorphenamine Maleate/Caffeine/SulfogaiacolApprovedMainland ChinaCommon ColdZhejiang Apeloa Kangyu Pharmaceutical Co Ltd
Common Cold
Details
Dextromethorphan Hydrobromide/Chlorphenamine Maleate/Sodium Citrate/Ammonium Chloride/CaffeineApproved尔可芬
Cough
Details
Acetaminophen/Caffeine/Codeine Phosphate/Diphenhydramine HydrochlorideApproved斯力帮
Headache
Details
Ferric Ammonium Citrate/Vitamin B1/Sodium glycerophosphate/CaffeineApproved
Ischemia
Details
Norethidranum Dipropionas/Caffeine/Vitamin B6ApprovedMainland ChinaContraceptionHuazhong Pharmaceutical Co Ltd1981-01-01
Contraception
Details
Acetaminophen/Propyphenazone/CaffeineApproved散利痛, 散列通
Common Cold
Details
Quinine Hydrochloride Hydrate/CaffeineApproved
Malaria
Details
Dihydroergocryptine/CaffeineApproved洛斯宝, VASOBRAL
Diabetes Mellitus; Diabetic Retinopathy
Details
Aminophenazone/Phenacetin/CaffeineApproved
Fever; Pain
Details
Aminophenazone/Caffeine/Calcium GlycerophosphateApproved
Dysmenorrhea; Headache; Neuralgia
Details
Acetaminophen/Caffeine/Chlorphenamine MaleateApproved
Common Cold
Details
Aminophenazone/Caffeine/Chlorphenamine MaleateApproved
Common Cold; Headache; Neuralgia
Details
Aspirin/Caffeine/Codeine PhosphateApproved柯克
Pain
Details
Acetaminophen/Pseudoephedrine Hydrochloride/CaffeineApproved
Common Cold
Details
Aspirin/Acetaminophen/Caffeine/Chlorphenamine MaleateApproved
Common Cold
Details
Aspirin/Caffeine/Chlorphenamine Maleate/Tartaric AcidApproved
Common Cold
Details
Acetaminophen/Caffeine/Pseudoephedrine Hydrochloride/Chlorphenamine MaleateApproved
Common Cold
Details
Aminophenazone/Phenacetin/Caffeine/PhenobarbitalApproved
Migraine Disorders
Details
Acetaminophen/Chlorphenamine Maleate/Caffeine/GuaifenesinApproved
Common Cold
Details
Acetaminophen/Amantadine Hydrochloride/Caffeine/Artificial BezoarApproved
Common Cold
Details
Acetaminophen/Salicylamide/Pseudoephedrine Hydrochloride/Caffeine/Triprolidine Hydrochloride HydrateApproved联邦菲迪乐
Common Cold
Details
Sodium Benzoate/CaffeineApproved
Central Nervous System Diseases
Details
Aminophenazone/CaffeineApproved
Fever
Details
Antipyrine/CaffeineApproved
Common Cold
Details
Aspirin/CaffeineApproved
Common Cold
Details
Antipyrine/Caffeine/Citric AcidApproved米格来宁Mainland ChinaSedationMudanjiang Lingtai Medicdment Co Ltd, Xi'An Disai Biological Pharmaceutical Co Ltd, Heilongjiang Hasing Pharmaceutical Group Co Ltd, Huadong Medicine (Xi'An) Bodyguard Pharmaceutical Co Ltd1982-01-01
Sedation
Details
Aminophenazone/Acetaminophen/Caffeine/Chlorphenamine MaleateApproved克感敏, 扑感敏, 朴感敏
Common Cold
Details
Acetaminophen/Caffeine/Ephedrine Hydrochloride/Diphenhydramine HydrochlorideApproved
Influenza, Human
Details
Acetaminophen/Caffeine/Chlorphenamine Maleate/Artificial BezoarApproved
Common Cold
Details
Aspirin/Phenacetin/CaffeineApproved
Arthralgia; Dysmenorrhea; Fever; Headache; Neuralgia; Toothache
Details
Aspirin/Caffeine/AcetaminophenApprovedUnited StatesMigraine DisordersHaleon PLC
Anesthesia; Migraine Disorders
Details
Acetaminophen/Butalbital/CaffeineApproved
Headache
Details
Acetaminophen/CaffeineApprovedZentiva AsMainland ChinaPainSino--American Shanghai Squibb Pharmaceutical Ltd
Pain
Details
Sodium glycerophosphate/Caffeine/Vitamin B/Phosphoric Acid/NiacinApproved
Details
Acetaminophen/Caffeine/Phenylephrine Hydrochloride/Chlorphenamine Maleate/Vitamin BApproved
Details
Acetaminophen/Chlorphenamine Maleate/Methylephedrine Hydrochloride/Sulfogaiacol/CaffeineApprovedMainland ChinaCommon ColdHainan Sanfengyou Pharmaceutical Co Ltd2006-05-16
Common Cold
Details
Brompheniramine Maleate/Bromhexine Hydrochloride/Caffeine/Acetaminophen/Phenylephrine HydrochlorideApproved
Common Cold
Details
Acetaminophen/Amantadine Hydrochloride/Caffeine/Chlorphenamine Maleate/Artificial BezoarApproved复方氨酚烷胺Mainland ChinaCommon Coldnull1984-01-01
Common Cold
Details
CaffeineApproved
Apnea; Cocaine-Related Disorders; Cognitive Dysfunction; Consciousness; Delirium; Diabetes Complications; Diabetes Mellitus, Type 1; Diabetic Nephropathies; Disorders of Excessive Somnolence; Fatigue; Fetal Membranes, Premature Rupture; Intermittent Claudication; Memory Disorders; Mental Fatigue; Parkinson Disease; Postoperative Cognitive Complications; Sexual Dysfunction, Physiological; Sleepiness; Spinal Cord Injuries
Details
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